Belinostat
CAS No. 414864-00-9
Belinostat ( PXD101 )
Catalog No. M14420 CAS No. 414864-00-9
Belinostat is a novel hydroxamic acid-type histone deacetylase (HDAC) inhibitor with antineoplastic activity.
Purity : >98%(HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
Size | Price / USD | Stock | Quantity |
5MG | 35 | In Stock |
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10MG | 56 | In Stock |
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25MG | 88 | In Stock |
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50MG | 132 | In Stock |
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100MG | 195 | In Stock |
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200MG | 312 | In Stock |
|
500MG | 520 | In Stock |
|
1G | Get Quote | In Stock |
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Biological Information
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Product NameBelinostat
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NoteResearch use only, not for human use.
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Brief DescriptionBelinostat is a novel hydroxamic acid-type histone deacetylase (HDAC) inhibitor with antineoplastic activity.
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DescriptionBelinostat is a novel hydroxamic acid-type histone deacetylase (HDAC) inhibitor with antineoplastic activity. Belinostat targets HDAC enzymes, thereby inhibiting tumor cell proliferation, inducing apoptosis, promoting cellular differentiation, and inhibiting angiogenesis. This agent may sensitize drug-resistant tumor cells to other antineoplastic agents, possibly through a mechanism involving the down-regulation of thymidylate synthase.
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SynonymsPXD101
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PathwayCell Cycle/DNA Damage
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TargetHDAC
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RecptorHDAC
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Research AreaCancer
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Indication——
Chemical Information
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CAS Number414864-00-9
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Formula Weight318.35
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Molecular FormulaC15H14N2O4S
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Purity>98%(HPLC)
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SolubilityDMSO: 64 mg/mL (201.03 mM)
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SMILESC1=CC=C(C=C1)NS(=O)(=O)C2=CC=CC(=C2)/C=C/C(=O)NO
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Chemical Name2-Propenamide, N-hydroxy-3-(3-((phenylamino)sulfonyl)phenyl)-
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Savickiene J, et al. anticancer Drugs. 2014 Sep;25(8):938-49.
molnova catalog
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